.Pharmacolibrary.Drugs.ATC.B.B01AC56

Information

name:AcetylsalicylicAcidCombinationsWithProtonPumpInhibitors
ATC code:B01AC56
route:oral
compartments:1
dosage:100mg
volume of distribution:11L
clearance:37L/h
other parameters in model implementation

Acetylsalicylic acid (ASA), commonly known as aspirin, is an antiplatelet medication used widely for secondary prevention of cardiovascular events (such as heart attack or stroke). It is sometimes combined with proton pump inhibitors (PPIs) to reduce the risk of gastrointestinal side effects, particularly gastrointestinal bleeding, in patients requiring long-term ASA therapy. This combination is approved and used today for cardiovascular protection in at-risk populations.

Pharmacokinetics

Pharmacokinetic parameters are estimated for healthy adults administered oral fixed-dose acetylsalicylic acid/proton pump inhibitor combination.

References

  1. Echizen, H (2016). The First-in-Class Potassium-Competitive Acid Blocker, Vonoprazan Fumarate: Pharmacokinetic and Pharmacodynamic Considerations. Clinical pharmacokinetics 55(4) 409–418. DOI:10.1007/s40262-015-0326-7 PUBMED:https://pubmed.ncbi.nlm.nih.gov/26369775

Revisions


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