name: | Lomitapide |
ATC code: | C10AX12 | route: | oral |
n-compartments | 1 |
Lomitapide is a microsomal triglyceride transfer protein (MTP) inhibitor used as an adjunct treatment for lowering low-density lipoprotein cholesterol (LDL-C) levels in patients with homozygous familial hypercholesterolemia (HoFH). It is approved for use in adults as an adjunct to other lipid-lowering therapies and dietary modifications.
Pharmacokinetic parameters for lomitapide in healthy adults after oral administration under fasting conditions.