.Pharmacolibrary.Drugs.ATC.N.N01AH06

Information

name:Remifentanil
ATC code:N01AH06
route:intravenous
n-compartments3

Remifentanil is an ultra-short-acting synthetic opioid analgesic approved for use as an adjunct to anesthesia during surgery or for sedation in intensive care settings. It is administered intravenously due to its rapid hydrolysis by nonspecific blood and tissue esterases, which gives it a very short context-sensitive half-life. Remifentanil is widely used in clinical practice today for its predictable, rapid onset and offset.

Pharmacokinetics

Pharmacokinetic parameters in healthy adult volunteers administered intravenous remifentanil (aged 19–53 years, both sexes).

References

  1. Ziesenitz, VC, et al., & van den Anker, JN (2018). Pharmacokinetics of Fentanyl and Its Derivatives in Children: A Comprehensive Review. Clinical pharmacokinetics 57(2) 125–149. DOI:10.1007/s40262-017-0569-6 PUBMED:https://pubmed.ncbi.nlm.nih.gov/28688027

  2. Imaizumi, T, et al., & Murakawa, M (2017). Population pharmacokinetics of intravenous acetaminophen in Japanese patients undergoing elective surgery. Journal of anesthesia 31(3) 380–388. DOI:10.1007/s00540-017-2358-7 PUBMED:https://pubmed.ncbi.nlm.nih.gov/28432468

  3. Kamata, M, & Tobias, JD (2016). Remifentanil: applications in neonates. Journal of anesthesia 30(3) 449–460. DOI:10.1007/s00540-015-2134-5 PUBMED:https://pubmed.ncbi.nlm.nih.gov/26758072

Revisions


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