.Pharmacolibrary.Drugs.ATC.N.N06AB06

Information

name:Sertraline
ATC code:N06AB06
route:oral
n-compartments2

Sertraline is a selective serotonin reuptake inhibitor (SSRI) antidepressant indicated for the treatment of major depressive disorder, obsessive-compulsive disorder, panic disorder, post-traumatic stress disorder, social anxiety disorder, and premenstrual dysphoric disorder. It is widely approved and used today in adults and pediatric patients for certain indications.

Pharmacokinetics

Pharmacokinetic parameters reported for healthy adult volunteers after oral administration of sertraline tablets.

References

  1. Alhadab, AA, & Brundage, RC (2020). Population Pharmacokinetics of Sertraline in Healthy Subjects: a Model-Based Meta-analysis. The AAPS journal 22(4) 73–None. DOI:10.1208/s12248-020-00455-y PUBMED:https://pubmed.ncbi.nlm.nih.gov/32430638

  2. Zang, YN, et al., & Ruan, CJ (2024). Population pharmacokinetics of olanzapine in pediatric patients with psychiatric disorders. Expert opinion on drug metabolism & toxicology 20(8) 827–840. DOI:10.1080/17425255.2024.2380472 PUBMED:https://pubmed.ncbi.nlm.nih.gov/39010781

  3. Wang, JH, et al., & Zhou, HH (2001). Pharmacokinetics of sertraline in relation to genetic polymorphism of CYP2C19. Clinical pharmacology and therapeutics 70(1) 42–47. DOI:10.1067/mcp.2001.116513 PUBMED:https://pubmed.ncbi.nlm.nih.gov/11452243

Revisions


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