.Pharmacolibrary.Drugs.ATC.R.R05CB01_1

Information

name:Acetylcysteine_1
ATC code:R05CB01_1
route:intravenous
n-compartments2

Acetylcysteine (N-acetylcysteine, NAC) is a mucolytic agent used to break down mucus, particularly in the lungs. It is also used as an antidote for acetaminophen (paracetamol) overdose. Approved and widely used in clinical practice today.

Pharmacokinetics

Pharmacokinetic parameters in patients after intravenous administration of NAC for acetaminophen overdose (standard 21-hour protocol).

References

  1. Forrest, JA, et al., & Prescott, LF (1982). Clinical pharmacokinetics of paracetamol. Clinical pharmacokinetics 7(2) 93–107. DOI:10.2165/00003088-198207020-00001 PUBMED:https://pubmed.ncbi.nlm.nih.gov/7039926

  2. Anderson, SM, et al., & Patel, RV (2011). Intravenous N-acetylcysteine in the prevention of contrast media-induced nephropathy. The Annals of pharmacotherapy 45(1) 101–107. DOI:10.1345/aph.1P275 PUBMED:https://pubmed.ncbi.nlm.nih.gov/21205947

  3. Fayed, MS, et al., & Coles, LD (2023). Population Pharmacokinetic Model of N-Acetylcysteine During Periods of Recurrent Hypoglycemia in Healthy Volunteers. Clinical pharmacology in drug development 12(12) 1234–1240. DOI:10.1002/cpdd.1338 PUBMED:https://pubmed.ncbi.nlm.nih.gov/37937383

Revisions


Generated at 2025-07-21T18:21:10Z by OpenModelicaOpenModelica 1.25.1 using GenerateDoc.mos