.Pharmacolibrary.Drugs.ATC.V.V10XX05

Information

name:Lutetium177luVipivotideTetraxetan
ATC code:V10XX05
route:intravenous
n-compartments2

Lutetium (177Lu) vipivotide tetraxetan (INN; formerly known as lutetium-177 PSMA-617, trade name Pluvicto) is a radioligand therapeutic used for the treatment of prostate-specific membrane antigen (PSMA)-positive metastatic castration-resistant prostate cancer (mCRPC). Administered intravenously, it delivers targeted radiation to PSMA-expressing cancer cells. It is approved for clinical use in certain advanced prostate cancers.

Pharmacokinetics

Pharmacokinetic parameters reported in adult male patients with PSMA-positive metastatic castration-resistant prostate cancer following intravenous administration.

References

    Revisions


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