.Pharmacolibrary.Drugs.A_AlimentaryTractAndMetabolism.A01A_StomatologicalPreparations.A01AB04_AmphotericinB.AmphotericinB

Information

name:AmphotericinB
ATC code:A01AB04
route:intravenous
n-compartments2

Amphotericin B is a polyene antifungal agent primarily used for the treatment of serious systemic fungal infections, including aspergillosis, cryptococcosis, histoplasmosis, and candidiasis. It is generally reserved for severe cases due to its toxicity. Amphotericin B is approved for medical use and remains in clinical use, mainly as intravenous administration in hospital settings.

Pharmacokinetics

Pharmacokinetic parameters reported for adult patients with systemic fungal infections, following intravenous administration.

References

  1. Groll, AH, et al., & Brüggemann, RJM (2019). Clinical Pharmacokinetics, Pharmacodynamics, Safety and Efficacy of Liposomal Amphotericin B. Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 68(Suppl 4) S260–S274. DOI:10.1093/cid/ciz076 PUBMED:https://pubmed.ncbi.nlm.nih.gov/31222253

  2. Würthwein, G, et al., & Walsh, TJ (2005). Population pharmacokinetics of amphotericin B lipid complex in neonates. Antimicrobial agents and chemotherapy 49(12) 5092–5098. DOI:10.1128/AAC.49.12.5092-5098.2005 PUBMED:https://pubmed.ncbi.nlm.nih.gov/16304177

  3. Nath, CE, et al., & Earl, JW (2001). Population pharmacokinetics of amphotericin B in children with malignant diseases. British journal of clinical pharmacology 52(6) 671–680. DOI:10.1046/j.0306-5251.2001.01496.x PUBMED:https://pubmed.ncbi.nlm.nih.gov/11736878

Revisions


Generated at 2025-07-21T18:21:10Z by OpenModelicaOpenModelica 1.25.1 using GenerateDoc.mos