.Pharmacolibrary.Drugs.A_AlimentaryTractAndMetabolism.A01A_StomatologicalPreparations.A01AC04_Prednisolone.Prednisolone

Information

name:Prednisolone
ATC code:A01AC04
route:oral
n-compartments2

Prednisolone is a synthetic glucocorticoid and anti-inflammatory agent widely used in the treatment of a variety of conditions including asthma, rheumatoid arthritis, autoimmune disorders, inflammatory diseases, and allergies. It is an active metabolite of prednisone and is approved and in common clinical use today.

Pharmacokinetics

Pharmacokinetic parameters for healthy adult volunteers after a single oral dose.

References

  1. de Truchis, C, et al., & Boyer, O (2023). Prednisolone pharmacokinetics after oral prednisone administration in paediatric patients with kidney transplant. British journal of clinical pharmacology 89(5) 1532–1540. DOI:10.1111/bcp.15610 PUBMED:https://pubmed.ncbi.nlm.nih.gov/36510685

  2. Petersen, KB, et al., & Schmiegelow, K (2003). Population pharmacokinetics of prednisolone in children with acute lymphoblastic leukemia. Cancer chemotherapy and pharmacology 51(6) 465–473. DOI:10.1007/s00280-003-0602-3 PUBMED:https://pubmed.ncbi.nlm.nih.gov/12698270

  3. Yoshida, K, et al., & Chanu, P (2021). Population Pharmacokinetics of Ipatasertib and Its Metabolite in Cancer Patients. Journal of clinical pharmacology 61(12) 1579–1591. DOI:10.1002/jcph.1942 PUBMED:https://pubmed.ncbi.nlm.nih.gov/34273118

Revisions


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