.Pharmacolibrary.Drugs.A_AlimentaryTractAndMetabolism.A02B_DrugsForPepticUlcerAndGastroOesophagealRefluxDis.A02BC53_LansoprazoleCombinations.LansoprazoleCombinations

Information

name:LansoprazoleCombinations
ATC code:A02BC53
route:oral
n-compartments2

Lansoprazole, in combination formulations (ATC: A02BC53), is a proton pump inhibitor used to treat conditions like gastroesophageal reflux disease (GERD), peptic ulcer disease, and Zollinger–Ellison syndrome where reduction of gastric acid secretion is desired. Combination products may include antimicrobials, such as those for Helicobacter pylori eradication, or other agents for gastrointestinal protection. Lansoprazole is approved and widely used today either alone or in such combinations.

Pharmacokinetics

Estimated pharmacokinetic parameters for an adult population administered lansoprazole combinations orally; no combination-specific PK literature available, values estimated based on single oral lansoprazole PK data in healthy adults.

References

  1. Echizen, H (2016). The First-in-Class Potassium-Competitive Acid Blocker, Vonoprazan Fumarate: Pharmacokinetic and Pharmacodynamic Considerations. Clinical pharmacokinetics 55(4) 409–418. DOI:10.1007/s40262-015-0326-7 PUBMED:https://pubmed.ncbi.nlm.nih.gov/26369775

  2. Litalien, C, et al., & Faure, C (2005). Pharmacokinetics of proton pump inhibitors in children. Clinical pharmacokinetics 44(5) 441–466. DOI:10.2165/00003088-200544050-00001 PUBMED:https://pubmed.ncbi.nlm.nih.gov/15871633

  3. Yu, L, et al., & Zhang, Y (2023). Pharmacokinetics and Pharmacodynamics of Lansoprazole/Sodium Bicarbonate Immediate-release Capsules in Healthy Chinese Subjects: An Open, Randomized, Controlled, Crossover, Single-, and Multiple-dose Trial. Clinical pharmacology in drug development 12(9) 902–910. DOI:10.1002/cpdd.1251 PUBMED:https://pubmed.ncbi.nlm.nih.gov/37165834

Revisions


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