.Pharmacolibrary.Drugs.A_AlimentaryTractAndMetabolism.A07E_IntestinalAntiinflammatoryAgents.A07EA03_Prednisone.Prednisone

Information

name:Prednisone
ATC code:A07EA03
route:oral
n-compartments1

Prednisone is a synthetic glucocorticoid drug commonly used as an anti-inflammatory and immunosuppressant in the treatment of conditions such as asthma, rheumatoid arthritis, allergic disorders, and autoimmune diseases. It is an oral prodrug, metabolized in the liver to its active form, prednisolone. Prednisone is widely approved and used in clinical practice today.

Pharmacokinetics

Pharmacokinetic parameters reported for healthy adult volunteers after oral administration.

References

  1. de Truchis, C, et al., & Boyer, O (2023). Prednisolone pharmacokinetics after oral prednisone administration in paediatric patients with kidney transplant. British journal of clinical pharmacology 89(5) 1532–1540. DOI:10.1111/bcp.15610 PUBMED:https://pubmed.ncbi.nlm.nih.gov/36510685

  2. Romano-Aguilar, M, et al., & Romano-Moreno, S (2020). Population pharmacokinetics of mycophenolic acid in Mexican patients with lupus nephritis. Lupus 29(9) 1067–1077. DOI:10.1177/0961203320931567 PUBMED:https://pubmed.ncbi.nlm.nih.gov/32539658

  3. Velickovic-Radovanovic, R, et al., & Jankovic, SM (2010). Population pharmacokinetics of tacrolimus in kidney transplant patients. International journal of clinical pharmacology and therapeutics 48(6) 375–382. DOI:10.5414/cpp48375 PUBMED:https://pubmed.ncbi.nlm.nih.gov/20497746

Revisions


Generated at 2025-07-21T18:21:10Z by OpenModelicaOpenModelica 1.25.1 using GenerateDoc.mos