.Pharmacolibrary.Drugs.A_AlimentaryTractAndMetabolism.A07E_IntestinalAntiinflammatoryAgents.A07EA06_Budesonide.Budesonide

Information

name:Budesonide
ATC code:A07EA06
route:oral
n-compartments2

Budesonide is a glucocorticoid steroid with potent anti-inflammatory properties. It is primarily used in the treatment of inflammatory bowel diseases, such as Crohn's disease and ulcerative colitis, and is approved for oral and inhaled use in numerous countries. It has a significant first-pass metabolism, limiting its systemic effects.

Pharmacokinetics

Pharmacokinetic parameters reported in healthy adult volunteers after oral administration.

References

  1. Simeoli, R, et al., & Goffredo, BM (2024). Pharmacokinetic Evaluation of Oral Viscous Budesonide in Paediatric Patients with Eosinophilic Oesophagitis in Repaired Oesophageal Atresia. Pharmaceutics 16(7) –. DOI:10.3390/pharmaceutics16070872 PUBMED:https://pubmed.ncbi.nlm.nih.gov/39065569

  2. Donnelly, R, & Seale, JP (2001). Clinical pharmacokinetics of inhaled budesonide. Clinical pharmacokinetics 40(6) 427–440. DOI:10.2165/00003088-200140060-00004 PUBMED:https://pubmed.ncbi.nlm.nih.gov/11475468

  3. Abdalla, MI, & Herfarth, H (2016). Budesonide for the treatment of ulcerative colitis. Expert opinion on pharmacotherapy 17(11) 1549–1559. DOI:10.1080/14656566.2016.1183648 PUBMED:https://pubmed.ncbi.nlm.nih.gov/27157244

Revisions


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