.Pharmacolibrary.Drugs.A_AlimentaryTractAndMetabolism.A10B_BloodGlucoseLoweringDrugsExclInsulins.A10BB06_Carbutamide.Carbutamide

Information

name:Carbutamide
ATC code:A10BB06
route:oral
n-compartments1

Carbutamide is a first-generation sulfonylurea oral hypoglycemic drug historically used to treat type 2 diabetes mellitus. It acts by stimulating insulin secretion from pancreatic beta-cells. Carbutamide is largely obsolete and is not commonly used in clinical practice today due to safer alternatives with better efficacy and lower risk of adverse effects.

Pharmacokinetics

Pharmacokinetic parameters estimated for a typical adult (based on pharmacological class analogs and limited historical data). No recent or direct human PK studies with full parameterization are available for carbutamide.

References

    Revisions


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