.Pharmacolibrary.Drugs.B_BloodAndBloodFormingOrgans.B01A_AntithromboticAgents.B01AX05_Fondaparinux.Fondaparinux

Information

name:Fondaparinux
ATC code:B01AX05
route:subcutaneous
n-compartments1

Fondaparinux is a synthetic pentasaccharide anticoagulant that selectively inhibits Factor Xa via antithrombin III. It is used for the prevention and treatment of deep vein thrombosis (DVT) and pulmonary embolism (PE), particularly after orthopedic surgery. Fondaparinux is approved and currently used in clinical practice.

Pharmacokinetics

Pharmacokinetic parameters in healthy adult volunteers after subcutaneous administration.

References

  1. Hanada, K, et al., & Takahashi, H (2018). Population pharmacokinetics and pharmacodynamics of fondaparinux in Japanese patients after artificial total knee replacement
. International journal of clinical pharmacology and therapeutics 56(6) 255–262. DOI:10.5414/CP203169 PUBMED:https://pubmed.ncbi.nlm.nih.gov/29595122

  2. Bauer, KA, et al., & Meuleman, DG (2002). Fondaparinux, a synthetic pentasaccharide: the first in a new class of antithrombotic agents - the selective factor Xa inhibitors. Cardiovascular drug reviews 20(1) 37–52. DOI:10.1111/j.1527-3466.2002.tb00081.x PUBMED:https://pubmed.ncbi.nlm.nih.gov/12070533

  3. Gerotziafas, GT, et al., & Elalamy, I (2014). New orally active anticoagulant agents for the prevention and treatment of venous thromboembolism in cancer patients. Therapeutics and clinical risk management 10 423–436. DOI:10.2147/TCRM.S49063 PUBMED:https://pubmed.ncbi.nlm.nih.gov/24966680

Revisions


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