.Pharmacolibrary.Drugs.C_CardiovascularSystem.C10A_LipidModifyingAgentsPlain.C10AB04_Gemfibrozil.Gemfibrozil

Information

name:Gemfibrozil
ATC code:C10AB04
route:oral
n-compartments1

Gemfibrozil is a lipid-regulating drug classified as a fibric acid derivative, used primarily for the treatment of hyperlipidemia and hypertriglyceridemia. It is indicated to reduce cardiovascular risk in dyslipidemic patients, particularly those with high triglycerides. Gemfibrozil is still approved and in clinical use today.

Pharmacokinetics

Pharmacokinetic parameters in healthy adult volunteers after oral administration under fasting conditions.

References

  1. Bi, YA, et al., & Varma, MVS (2024). Mechanistic Determinants of Daprodustat Drug-Drug Interactions and Pharmacokinetics in Hepatic Dysfunction and Chronic Kidney Disease: Significance of OATP1B-CYP2C8 Interplay. Clinical pharmacology and therapeutics 115(6) 1336–1345. DOI:10.1002/cpt.3215 PUBMED:https://pubmed.ncbi.nlm.nih.gov/38404228

  2. Plosker, GL, & Figgitt, DP (2004). Repaglinide : a pharmacoeconomic review of its use in type 2 diabetes mellitus. PharmacoEconomics 22(6) 389–411. DOI:10.2165/00019053-200422060-00005 PUBMED:https://pubmed.ncbi.nlm.nih.gov/15099124

  3. Maher, S, et al., & Hayden, JC (2019). Effect of Overencapsulation on the Disintegration and Dissolution of Licensed Formulations for Blinding in Randomized Controlled Trials. Journal of pharmaceutical sciences 108(3) 1227–1235. DOI:10.1016/j.xphs.2018.10.035 PUBMED:https://pubmed.ncbi.nlm.nih.gov/30385287

Revisions


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