.Pharmacolibrary.Drugs.H_SystemicHormonalPreparationsExclSexHormonesAndInsulins.H02A_CorticosteroidsForSystemicUsePlain.H02AB04_Methylprednisolone.Methylprednisolone_1

Information

name:Methylprednisolone_1
ATC code:H02AB04_1
route:oral
n-compartments1

Methylprednisolone is a synthetic glucocorticoid corticosteroid drug with potent anti-inflammatory and immunosuppressive properties. It is widely used to treat conditions such as allergic reactions, autoimmune diseases, certain types of arthritis, and is also employed in transplant rejection prophylaxis. It is approved and commonly used in clinical practice today.

Pharmacokinetics

Pharmacokinetic parameters after single oral dose in healthy adult male volunteers.

References

  1. Wang, DD, et al., & Li, ZP (2018). Population pharmacokinetics of tacrolimus in paediatric systemic lupus erythematosus based on real-world study. Journal of clinical pharmacy and therapeutics 43(4) 476–483. DOI:10.1111/jcpt.12707 PUBMED:https://pubmed.ncbi.nlm.nih.gov/29766530

  2. Tornatore, KM, et al., & Venuto, RC (1995). Methylprednisolone pharmacokinetics, cortisol response, and adverse effects in black and white renal transplant recipients. Transplantation 59(5) 729–736. DOI:10.1097/00007890-199503150-00016 PUBMED:https://pubmed.ncbi.nlm.nih.gov/7886801

  3. Mehta, J, et al., & Kaushik, NK (2022). Role of Dexamethasone and Methylprednisolone Corticosteroids in Coronavirus Disease 2019 Hospitalized Patients: A Review. Frontiers in microbiology 13 813358–None. DOI:10.3389/fmicb.2022.813358 PUBMED:https://pubmed.ncbi.nlm.nih.gov/35242118

Revisions


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