.Pharmacolibrary.Drugs.J_AntiinfectivesForSystemicUse.J01E_SulfonamidesAndTrimethoprim.J01EB20_SulfonamidesInCombinatio.SulfonamidesInCombinatio

Information

name:SulfonamidesInCombination
ATC code:J01EB20
route:oral
n-compartments1

ATC code J01EB20 refers to combinations of short-acting sulfonamides, which are antibacterial agents primarily used in the past to treat urinary tract infections and other susceptible bacterial infections. Most sulfonamide combinations are not used widely today due to resistance and the development of newer antibiotics.

Pharmacokinetics

Estimated pharmacokinetic parameters for adult patients receiving oral sulfonamide combinations (e.g., sulfadiazine + sulfamerazine), as scientific publications with explicit population PK models for these combinations are lacking.

References

  1. Echizen, H (2016). The First-in-Class Potassium-Competitive Acid Blocker, Vonoprazan Fumarate: Pharmacokinetic and Pharmacodynamic Considerations. Clinical pharmacokinetics 55(4) 409–418. DOI:10.1007/s40262-015-0326-7 PUBMED:https://pubmed.ncbi.nlm.nih.gov/26369775

  2. Autmizguine, J, et al., & Gonzalez, D (2018). Population Pharmacokinetics of Trimethoprim-Sulfamethoxazole in Infants and Children. Antimicrobial agents and chemotherapy 62(1) –. DOI:10.1128/AAC.01813-17 PUBMED:https://pubmed.ncbi.nlm.nih.gov/29084742

  3. Suleiman, AA, et al., & Oberoi, RK (2020). Population Pharmacokinetics of Glecaprevir/Pibrentasvir in HCV-infected Japanese Subjects in Phase 3 CERTAIN-1 and CERTAIN-2 Trials. Journal of clinical pharmacology 60(3) 331–339. DOI:10.1002/jcph.1524 PUBMED:https://pubmed.ncbi.nlm.nih.gov/31515816

Revisions


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