.Pharmacolibrary.Drugs.J_AntiinfectivesForSystemicUse.J05A_DirectActingAntivirals.J05AE01_Saquinavir.Saquinavir_1 .Pharmacolibrary.Drugs.J_AntiinfectivesForSystemicUse.J05A_DirectActingAntivirals.J05AE01_Saquinavir.Saquinavir_1| name: | Saquinavir_1 |
| ATC code: | J05AE01_1 | route: | oral |
| n-compartments | 2 |
Saquinavir is a protease inhibitor used as an antiretroviral agent in the treatment of HIV-1 infection. It was one of the first protease inhibitors approved for use but is now less commonly used due to newer agents with improved safety and efficacy. It is used in combination antiretroviral therapy for managing HIV/AIDS.
Mean PK parameters in healthy volunteers after single 1200 mg oral dose of saquinavir (soft-gel capsule).
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