.Pharmacolibrary.Drugs.L_AntineoplasticAndImmunomodulatingAgents.L01E_ProteinKinaseInhibitors.L01EG02_Everolimus.Everolimus .Pharmacolibrary.Drugs.L_AntineoplasticAndImmunomodulatingAgents.L01E_ProteinKinaseInhibitors.L01EG02_Everolimus.Everolimus| name: | Everolimus |
| ATC code: | L01EG02 | route: | oral |
| n-compartments | 2 |
Everolimus is an orally available mTOR inhibitor used as an anticancer and immunosuppressive agent. It is indicated for the treatment of various cancers, including renal cell carcinoma, breast cancer, neuroendocrine tumors, as well as for prevention of organ transplant rejection. Everolimus is approved by regulatory agencies worldwide and in active clinical use today.
Pharmacokinetic parameters reported in adult cancer patients. Parameters reflect population pharmacokinetics after oral administration of 10 mg once daily.
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