.Pharmacolibrary.Drugs.L_AntineoplasticAndImmunomodulatingAgents.L01E_ProteinKinaseInhibitors.L01EN02_Pemigatinib.Pemigatinib .Pharmacolibrary.Drugs.L_AntineoplasticAndImmunomodulatingAgents.L01E_ProteinKinaseInhibitors.L01EN02_Pemigatinib.Pemigatinib| name: | Pemigatinib |
| ATC code: | L01EN02 | route: | oral |
| n-compartments | 2 |
Pemigatinib is an orally administered, selective inhibitor of fibroblast growth factor receptors (FGFR) 1, 2, and 3. It is primarily used in the treatment of cholangiocarcinoma (bile duct cancer) that is unresectable, locally advanced, or metastatic, specifically those with FGFR2 fusion or rearrangement. The drug is approved for clinical use in several regions including the US and EU.
Population pharmacokinetics in adult cancer patients, including cholangiocarcinoma, regardless of sex or age group, following oral administration.
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