.Pharmacolibrary.Drugs.L_AntineoplasticAndImmunomodulatingAgents.L04A_Immunosuppressants.L04AF01_Tofacitinib.Tofacitinib

Information

name:Tofacitinib
ATC code:L04AF01
route:oral
n-compartments2

Tofacitinib is an oral Janus kinase (JAK) inhibitor used for the treatment of autoimmune diseases such as rheumatoid arthritis, psoriatic arthritis, and ulcerative colitis. It is approved for use in adults and functions by modulating the immune response.

Pharmacokinetics

Healthy adult subjects, single-dose, oral administration.

References

  1. Vong, C, et al., & Mukherjee, A (2021). Population Pharmacokinetics of Tofacitinib in Patients With Moderate to Severe Ulcerative Colitis. Clinical pharmacology in drug development 10(3) 229–240. DOI:10.1002/cpdd.899 PUBMED:https://pubmed.ncbi.nlm.nih.gov/33513294

  2. Xie, R, et al., & Menon, S (2019). Population pharmacokinetics of tofacitinib in patients with psoriatic arthritis
. International journal of clinical pharmacology and therapeutics 57(9) 464–473. DOI:10.5414/CP203516 PUBMED:https://pubmed.ncbi.nlm.nih.gov/31319908

  3. Chang, C, et al., & Mukherjee, A (2024). Tofacitinib pharmacokinetics in children and adolescents with juvenile idiopathic arthritis. CPT: pharmacometrics & systems pharmacology 13(4) 599–611. DOI:10.1002/psp4.13104 PUBMED:https://pubmed.ncbi.nlm.nih.gov/38298058

Revisions


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