.Pharmacolibrary.Drugs.N_NervousSystem.N02A_Opioids.N02AB02_Pethidine.Pethidine_1

Information

name:Pethidine_1
ATC code:N02AB02_1
route:oral
n-compartments1

Pethidine (meperidine) is a synthetic opioid analgesic for moderate to severe pain, now rarely used due to side effect profile.

Pharmacokinetics

Pharmacokinetic parameters after oral administration in healthy adult volunteers.

References

  1. Forrest, JA, et al., & Prescott, LF (1982). Clinical pharmacokinetics of paracetamol. Clinical pharmacokinetics 7(2) 93–107. DOI:10.2165/00003088-198207020-00001 PUBMED:https://pubmed.ncbi.nlm.nih.gov/7039926

  2. Thigpen, JC, et al., & Harirforoosh, S (2019). Opioids: A Review of Pharmacokinetics and Pharmacodynamics in Neonates, Infants, and Children. European journal of drug metabolism and pharmacokinetics 44(5) 591–609. DOI:10.1007/s13318-019-00552-0 PUBMED:https://pubmed.ncbi.nlm.nih.gov/31006834

  3. Chan, K, et al., & Orme, ML (1990). Disposition of pethidine in man under acidic urinary pH. 4. Kinetics after oral dose in caucasian, Chinese and Indian subjects. Methods and findings in experimental and clinical pharmacology 12(1) 61–67. PUBMED:https://pubmed.ncbi.nlm.nih.gov/2314154

Revisions


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