.Pharmacolibrary.Drugs.P_AntiparasiticProductsInsecticidesAndRepellents.P02C_AntinematodalAgents.P02CA03_Albendazole.Albendazole

Information

name:Albendazole
ATC code:P02CA03
route:oral
n-compartments1

Albendazole is an anthelmintic drug used to treat a broad range of parasitic worm infestations, including neurocysticercosis, hydatid disease, giardiasis, and soil-transmitted helminthiases. It disrupts the microtubule formation in parasites, leading to their immobilization and death. Albendazole is widely approved and used globally for these indications.

Pharmacokinetics

Pharmacokinetic parameters reported in healthy adult volunteers after a single 400 mg oral dose, under fasting conditions.

References

  1. Whittaker, C, et al., & Boussinesq, M (2022). Factors associated with variation in single-dose albendazole pharmacokinetics: A systematic review and modelling analysis. PLoS neglected tropical diseases 16(10) e0010497–None. DOI:10.1371/journal.pntd.0010497 PUBMED:https://pubmed.ncbi.nlm.nih.gov/36306320

  2. Fimbo, AM, et al., & Aklillu, E (2023). Population pharmacokinetics of ivermectin after mass drug administration in lymphatic filariasis endemic communities of Tanzania. CPT: pharmacometrics & systems pharmacology 12(12) 1884–1896. DOI:10.1002/psp4.13038 PUBMED:https://pubmed.ncbi.nlm.nih.gov/37638539

  3. Pettarin, M, et al., & Kostewicz, ES (2020). A combined in vitro in-silico approach to predict the oral bioavailability of borderline BCS Class II/IV weak base albendazole and its main metabolite albendazole sulfoxide. European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences 155 105552–None. DOI:10.1016/j.ejps.2020.105552 PUBMED:https://pubmed.ncbi.nlm.nih.gov/32937212

Revisions


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