modelFolicAcid

Extends from Pharmacolibrary.Drugs.ATC.V.V04CX02.

Information

name:FolicAcid
ATC code:V04CX02
route:oral
compartments:1
dosage:400mg
volume of distribution:0.162L
clearance:7.0L/h
other parameters in model implementation

Folic acid is a water-soluble B-vitamin (vitamin B9) essential for DNA synthesis, repair, and methylation as well as amino acid metabolism. It is commonly used to prevent and treat folate deficiency, including megaloblastic anemia, and is recommended for women planning pregnancy to prevent neural tube defects. Folic acid is an approved and widely used drug.

Pharmacokinetics

Healthy adult volunteers, oral administration, fasting state.

References

  1. Lee, SK (2023). Issues of Women with Epilepsy and Suitable Antiseizure Drugs. Journal of epilepsy research 13(2) 23–35. DOI:10.14581/jer.23005 PUBMED:https://pubmed.ncbi.nlm.nih.gov/38223363

  2. Genton, P, et al., & Trinka, E (2006). Valproic acid in epilepsy : pregnancy-related issues. Drug safety 29(1) 1–21. DOI:10.2165/00002018-200629010-00001 PUBMED:https://pubmed.ncbi.nlm.nih.gov/16454531

  3. Bayes, J, et al., & Schloss, J (2019). The Bioavailability of Various Oral Forms of Folate Supplementation in Healthy Populations and Animal Models: A Systematic Review. Journal of alternative and complementary medicine (New York, N.Y.) 25(2) 169–180. DOI:10.1089/acm.2018.0086 PUBMED:https://pubmed.ncbi.nlm.nih.gov/30010385

Parameters

TypeNameDefaultDescription
Modelica.Units.SI.Massweight (from PK_1C)75patient weight (kg)
Modelica.Units.SI.SpecificVolumeVdPerKg (from PK_1C)0.9Volume of distribution (L/kg)
Modelica.Units.SI.MassFractionF (from PK_1C)0.8bioavailiability (0-1)
Pharmacolibrary.Types.ClearanceCl (from PK_1C)20clearance
Modelica.Units.SI.TimeadminTime (from PK_1C)60first administration time (s)
Modelica.Units.SI.TimeadminDuration (from PK_1C)600administration duration (s)
Modelica.Units.SI.TimeadminPeriod (from PK_1C)8*60*60period of administration (default 8 hours)(s)
Pharmacolibrary.Types.MassadminMass (from PK_1C)1000administration mass (mg)
IntegeradminCount (from PK_1C)8number of dose administered (1)
Pharmacolibrary.Types.VolumeVd (from PK_1C)VdPerKg*weightVolume of distribution (m3)
Pharmacolibrary.Types.MassConcentrationCmin (from PK_1C)0.004minimal therapeutic range
Pharmacolibrary.Types.MassConcentrationCmax (from PK_1C)0.008minimal therapeutic range
Pharmacolibrary.Types.MassConcentrationCtox_peak (from PK_1C)0.012toxicity peak level
Pharmacolibrary.Types.MassConcentrationCtox_trough (from PK_1C)0.006toxicity trough level
Pharmacolibrary.Types.TransferRateka (from PK_1C_enteral)0.016666666666666666first order absorption rate
Modelica.Units.SI.TimeTlag (from PK_1C_enteral)600delay between oral administration and absorption (default 10min)

Connectors

TypeNameDefaultDescription
Types.ConcentrationOutputC_central (from PK_1C)
Interfaces.ConcentrationPort_bcentralCPort (from PK_1C)

Components

TypeNameDefaultDescription
Pharmacokinetic.NoPerfusedTissueCompartmentcentral (from PK_1C)
Pharmacokinetic.ClearanceDrivenEliminationelim (from PK_1C)
Sources.PeriodicDoseperiodicDose (from PK_1C)
Modelica.Units.SI.Timet1_2 (from PK_1C)elimination half-life

Revisions

  • 06/2025 Tomas Kulhanek, generated model from data extracted from PUBMED, DrugBank and LLM(GPT4.1)