modelCarbonMonoxide

Extends from Pharmacolibrary.Drugs.ATC.V.V04CX08.

Information

name:CarbonMonoxide
ATC code:V04CX08
route:inhalation
compartments:1
dosage:30mg
volume of distribution:1L
clearance:0
other parameters in model implementation

Carbon monoxide is a colorless, odorless, and tasteless gas. In medical applications, it is used primarily as a diagnostic agent for measuring diffusing capacity of the lung (DLCO test) in pulmonary function testing, and experimentally as a research tool. It is not approved as a therapeutic drug but is administered under strict clinical conditions for diagnostic assessment. Carbon monoxide has high affinity for hemoglobin, displacing oxygen to form carboxyhemoglobin.

Pharmacokinetics

No published human pharmacokinetic model exists for carbon monoxide as a drug in standard clinical use. Carbon monoxide is typically administered by inhalation in diagnostic settings at very low concentrations (e.g., 0.3% in air, single breath or up to several minutes), and parameters such as absorption are governed by pulmonary uptake and binding to hemoglobin. No peer-reviewed publications were found providing compartment model parameters such as volume of distribution or clearance in the classic drug sense.

References

  1. Darby, TD, et al., & van Rossum, JM (1984). Cigarette smoking pharmacokinetics and its relationship to smoking behaviour. Clinical pharmacokinetics 9(5) 435–449. DOI:10.2165/00003088-198409050-00003 PUBMED:https://pubmed.ncbi.nlm.nih.gov/6388953

  2. Werley, MS, et al., & Lee, PN (2007). Possible effects on smokers of cigarette mentholation: a review of the evidence relating to key research questions. Regulatory toxicology and pharmacology : RTP 47(2) 189–203. DOI:10.1016/j.yrtph.2006.09.004 PUBMED:https://pubmed.ncbi.nlm.nih.gov/17097785

  3. Vélez de Mendizábal, N, et al., & Brown, JW (2015). Nicotine and cotinine exposure from electronic cigarettes: a population approach. Clinical pharmacokinetics 54(6) 615–626. DOI:10.1007/s40262-014-0221-7 PUBMED:https://pubmed.ncbi.nlm.nih.gov/25503588

Parameters

TypeNameDefaultDescription
Modelica.Units.SI.Massweight (from PK_1C)75patient weight (kg)
Modelica.Units.SI.SpecificVolumeVdPerKg (from PK_1C)0.9Volume of distribution (L/kg)
Modelica.Units.SI.MassFractionF (from PK_1C)0.8bioavailiability (0-1)
Pharmacolibrary.Types.ClearanceCl (from PK_1C)20clearance
Modelica.Units.SI.TimeadminTime (from PK_1C)60first administration time (s)
Modelica.Units.SI.TimeadminDuration (from PK_1C)600administration duration (s)
Modelica.Units.SI.TimeadminPeriod (from PK_1C)8*60*60period of administration (default 8 hours)(s)
Pharmacolibrary.Types.MassadminMass (from PK_1C)1000administration mass (mg)
IntegeradminCount (from PK_1C)8number of dose administered (1)
Pharmacolibrary.Types.VolumeVd (from PK_1C)VdPerKg*weightVolume of distribution (m3)
Pharmacolibrary.Types.MassConcentrationCmin (from PK_1C)0.004minimal therapeutic range
Pharmacolibrary.Types.MassConcentrationCmax (from PK_1C)0.008minimal therapeutic range
Pharmacolibrary.Types.MassConcentrationCtox_peak (from PK_1C)0.012toxicity peak level
Pharmacolibrary.Types.MassConcentrationCtox_trough (from PK_1C)0.006toxicity trough level

Connectors

TypeNameDefaultDescription
Types.ConcentrationOutputC_central (from PK_1C)
Interfaces.ConcentrationPort_bcentralCPort (from PK_1C)

Components

TypeNameDefaultDescription
Pharmacokinetic.NoPerfusedTissueCompartmentcentral (from PK_1C)
Pharmacokinetic.ClearanceDrivenEliminationelim (from PK_1C)
Sources.PeriodicDoseperiodicDose (from PK_1C)
Modelica.Units.SI.Timet1_2 (from PK_1C)elimination half-life

Revisions

  • 06/2025 Tomas Kulhanek, generated model from data extracted from PUBMED, DrugBank and LLM(GPT4.1)