.Pharmacolibrary.Drugs.N_NervousSystem.N05A_Antipsychotics.N05AH05_Asenapine.Asenapine

Information

Asenapine is an atypical antipsychotic drug indicated for the treatment of schizophrenia and bipolar disorder. It acts as an antagonist at multiple serotonergic, dopaminergic, and adrenergic receptors. It is approved and currently used as a sublingual or transdermal medication.

Pharmacokinetics

Healthy adult subjects, sublingual administration, single dose

References

1. Dogterom, P, et al., & Troyer, MD (2018). Asenapine pharmacokinetics and tolerability in a pediatric population. Drug design, development and therapy 12 2677–2693. DOI:10.2147/DDDT.S171475 PUBMED:https://pubmed.ncbi.nlm.nih.gov/30214156

Revisions

• 06/2025 initial generated model